Release Time:2019-03-11  Hits:

Indexed by: Journal Article

Date of Publication: 2017-11-17

Journal: ORGANIC LETTERS

Included Journals: PubMed、SCIE

Volume: 19

Issue: 22

Page Number: 6088-6091

ISSN: 1523-7060

Abstract: An efficient method for the synthesis of N-(quinolin-2-yl)sulfonamides is described. The intermolecular amidation of quinoline N-oxides with sulfonamides proceeded smoothly in the presence of PhI(OAc)(2) and PPh3 to afford N-(quinolin-2-yl)sulfonamides in satisfactory to excellent yields.