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Indexed by:期刊论文

Date of Publication:2010-01-01

Journal:JOURNAL OF HETEROCYCLIC CHEMISTRY

Included Journals:SCIE

Volume:47

Issue:1

Page Number:15-21

ISSN No.:0022-152X

Abstract:In recent years, protoporphyrinogen oxidase (Protox) inhibitor herbicides are developed rapidly, because of this type of herbicides shows high herbicidal activity and low toxicity. In this paper, we prepared a series of new substituted pyrazolyl benzoxazole derivative, which were synthesized from 4-fluorophenol, via a serial of reactions included chlorination, acylation, condensation, ring closure, methylation, nitration, and so on. All the structures are confirmed by (1)H NMR, MS and element analysis. Preliminary bioassay shows that most substituted pyrazolyl benzoxazole derivatives exhibit high herbicidal activity to the tested gramineous weeds and latifoliate weeds.