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Scientific Research
李悦青
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Associate Professor Supervisor of Master's Candidates
Scientific Research
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Li Haidong, Yao Qichao, Xu Feng, Li Yueqing, Kim Dayeh, Chung Jeewon, Baek Gain, Wu Xiaofeng, Hillman Prima Fitria, Lee Eun Young, Ge Haoying, Fan Jiangli, Wang Jingyun, Nam Sang-Jip, Peng Xiaojun, Yoon Juyoung.An Activatable AIEgen Probe for High-Fidelity Monitoring of Overexpressed Tumor Enzyme Activity and Its Application to Surgical Tumor Excision[J],Angewandte Chemie (International ed. in English),2020
Li, Guangzhe, Dong, Huijuan, Ma, Yao, Shao, Kun, Yueqing, Wu, Xiaodan, Yujie, Zhao, Weijie, Wang, SS (reprint author), Dalian Univ Technol, Dept Pharm, Sch Chem Engn, Dalian 116023, Peoples R China..Structure-activity relationships study of neolamellarin A and its analogues as hypoxia inducible factor-1 (HIF-1) inhibitors[J],BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,2019,29(16):2327-2331
Guo, Xiuhan, Li, Yueqing, Wang, Liu, Cai, Rui, Guangzhe, Zhao, Weijie, SS (reprint author), Dalian Univ Technol, Sch Pharmaceut Sci & Technol, Dalian 116023, Peoples R China., Wang, State Key Lab Fine Chem.Evaluation for in vitro Photodynamic Activity of Chlorin e(6)-Artesunate Conjugates by Irradiation with Different Wavelengths of Light Source[J],MACROHETEROCYCLES,2018,11(4):378-382
Li, Yue-qing, Dong, Yi, Ma, Xu, Hui-juan, Wu, Qian-qian, Zhao, Wei-jie, Guang-zhe.Orobanone analogues from acid-promoted aromatization rearrangement of curcumol inhibit hypoxia-inducible factor-1 (HIF-1) in cell-based reporter assays[J],BIOORGANIC CHEMISTRY,2019,85:357-363
Gao, Fengli, Li, Liuju, Fan, Jiangli, Cao, Jianfang, Yueqing, Chen, Liangyi, Peng, Xiaojun.An Off-On Two-Photon Carbazole-Based Fluorescent Probe: Highly Targeting and Super-Resolution Imaging of mtDNA[J],ANALYTICAL CHEMISTRY,2019,91(5):3336-3341
Wang, Shisheng, Liu, Liqiang, Guo, Xiuhan, Xu, Dong, Huijuan, Li, Yueqing, Zhao, Weijie, GZ (reprint author), Dalian Univ Technol, Sch Chem Engn, Dept Pharm, Dalian 116023, Peoples R China., Li, State Key Lab Fine Chem.Synthesis of novel natural product-like diaryl acetylenes as hypoxia inducible factor-1 inhibitors and antiproliferative agents[J],RSC ADVANCES,2019,9(24):13878-13886
Patents
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靶向Hsp60的黄酮烷氧基氨基磷酸酯衍生物、制备及应用
一种吡喃糖环吡咯螺缩酮生物碱的全合成方法及应用
一种应用近红外光谱法建立二维定性分析模型以鉴别鲜海刺参产地的方法
一类二氢卟吩半乳糖苷类化合物及其制备方法与应用
一类二氢卟吩葡萄糖苷类化合物及其制备方法与应用
具有光、声敏活性的二氢卟吩青蒿琥酯结合物及其制备方法与应用
Published Books
制药工程综合实验讲义
药物化学综合实验
Research Projects
基于低场核磁共振技术的药品品质分析的方法开发, 省、市、自治区科技项目, 2017/04/18-2023/09/13, 结题
基于吡咯螺缩酮生物碱仿生合成的小分子探针构建及抗衰老靶标蛋白的捕获, 国家自然科学基金项目, 2017/08/17, 结题
名优水产品品质溯源技术及监管体系研究与示范, 国家科技部, 2015/04/01, 结题
肿瘤低氧微环境选择性抗肿瘤活性化合物Furospinosulin-1的靶标蛋白发现用小分子探针的设计、合成与应用, 主管部门科技项目, 2015/03/02-2023/09/06, 结题
吡咯螺缩酮生物碱的仿生合成研究, 大连理工大学基本科研业务项目, 2019/03/25-2019/03/25, 在研
HIV-1 Vif-A3G相互作用的新型抑制剂的设计、合成与活性评价, 中央高校基本科研业务费专项, 2011/01/01-2012/12/31, 项目基于天然黄酮化合物的结构进行修饰和虚拟筛选,发现有潜力的化合物。